WebCytochrome P-450 CYP3A4 Inducers. All categories. Name Cytochrome P-450 CYP3A4 Inducers Accession Number ... Butalbital: A barbiturate drug used for symptomatic treatment of tension-type headache in various combinations with acetaminophen, aspirin, caffeine, and codeine. ... Cytochrome P450 3A4: enzyme: Enasidenib: UDP … WebOct 27, 2024 · The cytochrome P450 (CYP) enzyme family is the most important enzyme system catalyzing the phase 1 metabolism of pharmaceuticals and other xenobiotics such as herbal remedies and toxic compounds in the environment. The inhibition and induction of CYPs are major mechanisms causing pharmacokinetic drug–drug interactions. This …
Butalbital - Wikipedia
WebBarbiturates are enzyme inducers [98]. They induce CYP isoenzymes, such as the CYP2C and CYP3A families. Many interactions based on this mechanism have been described with phenobarbital, and would be expected to occur with other barbiturates. ... A possible interaction of imipramine with butalbital was reported in a 44-year-old woman, ... WebBupap (butalbital / acetaminophen) is a combination of two medications that help relieve different aspects of tension headaches. Tension headaches are commonly related to … bridge good to go fort atkinson
butalbital/acetaminophen/caffeine: Dosing ... - Epocrates
WebNifedipine is a CYP3A4 substrate and apalutamide is a strong CYP3A4 inducer. Coadministration of nifedipine with another strong CYP3A4 inducer reduced the AUC and Cmax of nifedipine by approximately 70%. Apomorphine: (Moderate) Use of calcium-channel blockers and apomorphine together can increase the hypotensive effects of … Web1 List of Herbal cytochrome P450 Inhibitors and Inducers. 2 See also. 3 Sources. Toggle the table of contents ... This is a list of cytochrome P450 modulators, or inhibitors and inducers of cytochrome P450 enzymes. Enzyme Inhibitors ... butalbital, phenobarbital) Capsaicin; Carbamazepine; Efavirenz; Enzalutamide; Glucocorticoids; Modafinil ... Webbutalbital/acetaminophen tablet 50mg/300mg (Orbivan CF) 50mg/325mg (Phrenilin) 50mg/650mg (Bupap) capsule 50mg/650mg (Phrenilin Forte) Tension Headache 1-2 tab/cap PO q4hr; not to exceed 6... bridge graphic organizer